SCHEMBL3632369

SCHEMBL3632369

CC(C)(C)N1CCC(Sc2cc(-c3cccc(C#N)c3)cc3ccncc23)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.40
VCP P55072 2/20 0.39
NEK1 Q96PY6 1/20 0.37
USP30 Q70CQ3 2/20 0.36
MAP4K1 Q92918 1/20 0.36
DHFR P00374 1/20 0.36
PDE4D Q08499 3/20 0.36
ROCK2 O75116 2/20 0.35
GRM5 P41594 1/20 0.35
CYP11B2 P19099 2/20 0.35
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
KMT2A Q03164 1/20 0.34
HIF1A Q16665 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13087449 0.85 CCNT1 (0.41) SLC22A12VCPMAP4K1DHFRCYP11B2
SCHEMBL2486778 0.85 GPR119 (0.45) SLC22A12
SCHEMBL2426906 0.84 CLK4 (0.42) SLC22A12VCPNEK1GRM5CYP11B2
SCHEMBL13090022 0.84 VCP (0.38) SLC22A12VCPNEK1USP30MAP4K1
SCHEMBL3630020 0.81 GPR6 (0.39) SLC22A12NEK1USP30MAP4K1PDE4D
SCHEMBL3628367 0.81 ROCK2 (0.47) SLC22A12NEK1MAP4K1ROCK2CYP1A2
SCHEMBL12327914 0.72 CYP11B1 (0.48) SLC22A12NEK1GRM5CYP11B2CYP17A1
SCHEMBL2424122 0.70 IKBKB (0.45) VCPNEK1PDE4DGRM5CYP11B2
SCHEMBL2492757 0.70 GPR119 (0.48) PDE4DPDE4APDE4BPDE4C
SCHEMBL2431769 0.69 CHRNB2 (0.51) SLC22A12NEK1GRM5CYP11B2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038465-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF 旭化成ファーマ株式会社 (JP) 2010-04-08 WO disclosed