SCHEMBL3633702

SCHEMBL3633702

O=CCc1cccnc1Nc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.51
MEN1 O00255 7/20 0.48
KMT2A Q03164 7/20 0.48
MAPT P10636 5/20 0.48
ALDH1A1 P00352 4/20 0.48
GAA P10253 1/20 0.48
GRM4 Q14833 1/20 0.42
RAB9A P51151 6/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
NPSR1 Q6W5P4 2/20 0.39
MAPK1 P28482 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
NPC1 O15118 4/20 0.38
HTT P42858 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1908379 0.81 DHODH (0.56) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL5252795 0.78 DHODH (0.51) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL9470451 0.78 DHODH (0.51) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL1375014 0.78 DHODH (0.56) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL2558369 0.77 NPC1 (0.41) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL25319320 0.75 MAPT (0.39) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL3634212 0.75 LMNA (0.42) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL14604182 0.75 DHODH (0.56) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL1376342 0.75 DHODH (0.56) DHODHMEN1KMT2AMAPTALDH1A1
SCHEMBL9753940 0.74 BRD4 (0.48) DHODHMEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694480-A1 ADAMANTYL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2014-02-12 EP disclosed
WO-2012136684-A1 ADAMANTYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2012-10-11 WO disclosed
EP-2148862-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. Hoffmann-Roche AG (CH) 2010-02-03 EP disclosed
WO-2009015917-A2 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed