SCHEMBL3634100

SCHEMBL3634100

COc1cc(Nc2nc3c(s2)CN(Cc2ccc(F)cc2)CC3)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
ABCB1 P08183 1/20 0.39
ALDH1A1 P00352 4/20 0.39
RAB9A P51151 4/20 0.39
MAPT P10636 4/20 0.39
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
GRM5 P41594 2/20 0.39
GRM1 Q13255 1/20 0.39
MEN1 O00255 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
GAA P10253 3/20 0.38
NPC1 O15118 2/20 0.38
MAPK1 P28482 1/20 0.38
MERTK Q12866 4/20 0.38
AXL P30530 1/20 0.38
MET P08581 1/20 0.38
ALOX15 P16050 1/20 0.37
LMNA P02545 1/20 0.37
GRIN1 Q05586 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636972 0.85 PSEN1 (0.40) KMT2AABCB1ALDH1A1RAB9AMAPT
SCHEMBL3642038 0.83 MKNK1 (0.41) KMT2AALDH1A1RAB9AMAPTKDM4E
SCHEMBL3636389 0.83 GRM5 (0.39) ABCB1RAB9AGRM5NPC1CDK9
SCHEMBL1036142 0.81 PSEN1 (0.54)
SCHEMBL3636592 0.81 GRM5 (0.34) KMT2AKDM4EGRM5GRM1ALOX15
SCHEMBL3639468 0.81 RAB9A (0.51) KMT2AALDH1A1RAB9AMAPTKDM4E
SCHEMBL3638385 0.80 NPC1 (0.40) ALDH1A1RAB9AGAANPC1ALOX15
SCHEMBL3633453 0.78 NPC1 (0.41) KMT2AALDH1A1RAB9AKDM4ESMN1; SMN2
SCHEMBL3638175 0.78 PSEN1 (0.36) ALDH1A1RAB9AKDM4EGAANPC1
SCHEMBL3636154 0.77 GRAMD1A (0.50) MAPTMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed