SCHEMBL3638385

SCHEMBL3638385

COc1cc(Nc2nc3c(s2)CN(S(C)(=O)=O)CC3)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
PSEN1 P49768 7/20 0.37
PSEN2 P49810 7/20 0.37
APH1B Q8WW43 7/20 0.37
NCSTN Q92542 7/20 0.37
APH1A Q96BI3 7/20 0.37
PSENEN Q9NZ42 7/20 0.37
ALOX15 P16050 1/20 0.36
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
PIK3CG P48736 2/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
JAK2 O60674 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3642038 0.88 MKNK1 (0.41) RAB9APSEN1PSEN2APH1BNCSTN
SCHEMBL3633453 0.88 NPC1 (0.41) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3638175 0.83 PSEN1 (0.36) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3639468 0.82 RAB9A (0.51) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3636154 0.82 GRAMD1A (0.50)
SCHEMBL1040137 0.81 PSEN1 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3636389 0.80 GRM5 (0.39) NPC1RAB9AROCK2ROCK1CYP1A2
SCHEMBL3636972 0.80 PSEN1 (0.40) NPC1RAB9APSEN1PSEN2APH1B
SCHEMBL3634100 0.80 KMT2A (0.40) NPC1RAB9AALOX15ALDH1A1LMNA
SCHEMBL3634269 0.80 PSEN1 (0.42) NPC1RAB9APSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed