SCHEMBL3634837

SCHEMBL3634837

[CH2]C(c1ccc2c(C)nccc2n1)N1CCN(S(=O)(=O)c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
EPHX2 P34913 1/20 0.44
GBA1 P04062 2/20 0.43
HSD11B1 P28845 2/20 0.43
TRPV4 Q9HBA0 2/20 0.43
GAA P10253 1/20 0.42
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 1/20 0.42
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
ATM Q13315 1/20 0.40
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
MAOA P21397 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633473 0.88 MEN1 (0.48) EPHX2GBA1MEN1KMT2A
SCHEMBL3633557 0.81 MEN1 (0.43) ALDH1A1GBA1GAAKDM4EMEN1
SCHEMBL3632513 0.79 CHRM1 (0.40) ALDH1A1GBA1HSD11B1MEN1KMT2A
SCHEMBL3632361 0.79 FPR2 (0.46) EPHX2
SCHEMBL3627516 0.78 ALDH1A1 (0.42) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL3321769 0.77 L3MBTL1 (0.49) ALDH1A1GBA1HSD11B1GAAKDM4E
SCHEMBL3634835 0.76 L3MBTL1 (0.46) ALDH1A1GBA1HSD11B1GAAKDM4E
SCHEMBL3633458 0.74 HRH3 (0.39) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL7682092 0.70 IKBKB (0.46) ALDH1A1EPHX2HSD11B1TRPV4GAA
SCHEMBL3632727 0.69 ACHE (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP claimed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO claimed
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP disclosed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO disclosed