SCHEMBL3633458

SCHEMBL3633458

[CH2]C(c1ccc2c(C)nccc2n1)N1CCN(c2ccc3c(C)nccc3n2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.39
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTR3A P46098 1/20 0.37
SORD Q00796 8/20 0.36
CYP1A2 P05177 3/20 0.36
USP2 O75604 2/20 0.36
EGFR P00533 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3663850 0.76 SIGMAR1 (0.45)
SCHEMBL3627516 0.75 ALDH1A1 (0.42) ALDH1A1KDM4ELMNASMN1; SMN2USP2
SCHEMBL3634837 0.74 ALDH1A1 (0.47) ALDH1A1KDM4EMEN1TSHRKMT2A
SCHEMBL3632727 0.73 ACHE (0.40) HRH3
SCHEMBL3633473 0.72 MEN1 (0.48) MEN1KMT2A
SCHEMBL3632361 0.71 FPR2 (0.46) HRH3
SCHEMBL3320791 0.71 HTR1A (0.43) HRH3ALDH1A1LMNAHTR3ACYP1A2
SCHEMBL3632513 0.70 CHRM1 (0.40) ALDH1A1MEN1KMT2A
SCHEMBL3633456 0.70 HRH3 (0.38) HRH3ALDH1A1HTR3ASORDCYP1A2
SCHEMBL3628240 0.63 ALDH1A1 (0.34) HRH3ALDH1A1KDM4EHTR3ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155748-A1 UROTENSIN II RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-02-24 EP claimed
WO-2008144268-A1 UROTENSIN II RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-27 WO claimed