Cadaverine Tartrate

Cadaverine Tartrate

SCHEMBL3634909

CS(=O)(=O)O.O=C(O)C(O)C(O)C(=O)O

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3CHRM1CHRM2CHRM3CHRM4ESR1ESR2GABRA1GABRB1GABRG2GBA1HRH1HTR1DHTR2AOPRD1OPRK1OPRM1SLC6A2SLC6A3TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cadaverine Tartrate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.32
ADRB2 known ✓ P07550 1/20 0.32
TSHR P16473 5/20 0.62
TP53 P04637 1/20 0.42
NFKB1 P19838 2/20 0.38
CYP2C19 P33261 1/20 0.38
CA2 P00918 1/20 0.35
CYP2C9 P11712 1/20 0.35
PDE4A P27815 1/20 0.35
PMP22 Q01453 2/20 0.34
TDP1 Q9NUW8 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HSD17B10 Q99714 2/20 0.32
BLM P54132 2/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
THPO P40225 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cadaverine Tartrate SCHEMBL988008 0.87 TSHR (0.71) TSHRTP53NFKB1CYP2C19CYP2C9
Cadaverine Tartrate SCHEMBL27906745 0.84 TSHR (0.67) TSHRTP53NFKB1CYP2C19CYP2C9
Cadaverine Tartrate SCHEMBL27547121 0.84 TSHR (0.67) TSHRTP53NFKB1CYP2C19CYP2C9
Cadaverine Tartrate SCHEMBL4193142 0.83 TSHR (0.43) TSHRTP53NFKB1CYP2C19TDP1
Cadaverine Tartrate SCHEMBL9345632 0.81 TSHR (0.62) TSHRTP53NFKB1CYP2C19CA2
Cadaverine Tartrate SCHEMBL9345627 0.81 TSHR (0.62) TSHRTP53NFKB1CYP2C19CA2
Cadaverine Tartrate SCHEMBL27491776 0.81 TSHR (0.62) TSHRTP53NFKB1CYP2C19CYP2C9
Cadaverine Tartrate SCHEMBL9437851 0.81 TSHR (0.62) TSHRTP53NFKB1CYP2C19CYP2C9
Cadaverine Tartrate SCHEMBL27906743 0.81 TSHR (0.62) TSHRTP53NFKB1CYP2C19CYP2C9
Lactic Acid SCHEMBL5538629 0.81 TP53 (0.69) TSHRTP53CYP2C19CA2PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030065173-A1 Pyridone-fused azabicyclic- or cytisine derivatives, their preparation and their use in addiction therapy O'NEILL BRIAN T (US) 2003-04-03 US claimed
WO-2024128359-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF BONE DISEASES 전남대학교산학협력단 2024-06-20 WO disclosed
WO-2024128335-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING BONE DISEASES 전남대학교산학협력단 2024-06-20 WO disclosed
CN-106890183-A A kind of dabigatran etcxilate pharmaceutical composition of high bioavilability 北京蓝丹医药科技有限公司 2017-06-27 CN disclosed
EP-2155719-A1 AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS Wyeth LLC (US) 2010-02-24 EP disclosed
WO-2008147945-A1 AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2008-12-04 WO disclosed
US-20080280981-A1 Tranexamic acid formulations XANODYNE PHARMACEUTICALS, INC. (US) 2008-11-13 US disclosed
US-20080146844-A1 PROCESS FOR PREPARING TOLTERODINE DR. REDDY'S LABORATORIES LIMITED (IN) 2008-06-19 US disclosed
US-7355077-B2 Process for preparing tolterodine DR. REDDY'S LABORATORIES LIMITED (IN) 2008-04-08 US disclosed
US-20060094904-A1 Reacting methyl 3-(2-benzyloxy-5-methyl phenyl)-3-phenylpropionate with a reducing agent to form 3-(2-benzyloxy-5-methylphenyl)-3-phenylpropanol DR. REDDY'S LABORATORIES LIMITED (IN) 2006-05-04 US disclosed
WO-1994014438-A1 HYDANTOIN AND SUCCINIMIDE-SUBSTITUTED DERIVATIVES OF SPIROINDANYLCAMPHORSULFONYL OXYTOCIN ANTAGONISTS MERCK & CO., INC. (US) 1994-07-07 WO disclosed
WO-1994007496-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-04-14 WO disclosed
WO-1993006092-A1 PIPERAZINYL (SULFONYL)AMIDE DERIVATIVES OF CAMPHOR AS OXYTOCIN ANTAGONISTS MERCK & CO., INC. (US) 1993-04-01 WO disclosed
CN-1070399-A The amide derivatives oxytocin antagonist that piperizinylcamphorsuoxytocin replaces MERCK & CO INC (US) 1993-03-31 CN disclosed
US-5137904-A Useful in the treatment of atherosclerosis and thrombosis G. D. SEARLE & CO. (US) 1992-08-11 US disclosed
EP-0486280-A2 Piperidinylcamphorsulfonyl oxytocin antagonists MERCK & CO. INC. (US) 1992-05-20 EP disclosed
WO-1992007821-A1 DIASTEREOISOMERS OF BICYCLO-SUBSTITUTED PHENYLACETONITRILE DERIVATIVES G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed
CN-87107723-A Agent of dihydropyridine anti-allergy and anti-inflammatory agent 1988-05-18 CN disclosed
US-4550105-A BETA-LACTAMASE INHIBITORS, ANTIBIOTICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-10-29 US disclosed
US-4547503-A 1-Cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-[4-(oxo-alkyl)-1-piperazinyl]quinoline-3-carboxylic acids and their derivatives, and antibacterial agents containing them BAYER AKTIENGESELLSCHAFT (DE) 1985-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080146844-A1 PROCESS FOR PREPARING TOLTERODINE ADRA2B, ADRB3, ADRB1 SLC6A2 814/4885ADRB2 5/4885TSHR 81/4885
US-20030065173-A1 Pyridone-fused azabicyclic- or cytisine derivatives, their preparation and their use in addiction therapy CHRNA5, CHRNA4, CHRNA10 SLC6A2 545/4885ADRB2 175/4885TSHR 2084/4885
US-20060094904-A1 Reacting methyl 3-(2-benzyloxy-5-methyl phenyl)-3-phenylpropionate with a reducing agent to form 3-(2-benzyloxy-5-methylphenyl)-3-phenylpropanol ADRB3, UGT1A3, COMT SLC6A2 500/4885ADRB2 18/4885TSHR 689/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.