SCHEMBL3635463

SCHEMBL3635463

CC(C)(C)OC(=O)N(Cc1ccccc1)S(=O)(=O)c1cccc(C#N)c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
STAT5B P51692 1/20 0.44
TAS2R14 Q9NYV8 2/20 0.44
HSD11B1 P28845 1/20 0.43
NR1H3 Q13133 1/20 0.41
ABCB1 P08183 1/20 0.41
CTSL P07711 2/20 0.41
CTSS P25774 2/20 0.41
MCOLN3 Q8TDD5 1/20 0.41
PTGES O14684 2/20 0.41
KCNH2 Q12809 1/20 0.41
CTSB P07858 1/20 0.40
GAA P10253 1/20 0.40
PTGER1 P34995 1/20 0.40
RORC P51449 1/20 0.40
NR1H2 P55055 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1857447 0.86 STAT5B (0.43) STAT5BTAS2R14HSD11B1CTSLCTSS
SCHEMBL1856320 0.85 STAT5B (0.42) STAT5BTAS2R14HSD11B1PTGESKCNH2
SCHEMBL1857129 0.83 STAT5B (0.46) STAT5BTAS2R14HSD11B1PTGESKCNH2
SCHEMBL28588131 0.79 TAS2R14 (0.55) STAT5BTAS2R14HSD11B1CTSLCTSS
SCHEMBL3724224 0.78 CA12 (0.43) STAT5BTAS2R14HSD11B1NR1H3RORC
SCHEMBL12550326 0.78 STAT5B (0.52) STAT5BTAS2R14HSD11B1PTGESKCNH2
SCHEMBL4925756 0.76 HTR2C (0.53) HSD11B1NR1H3MCOLN3
SCHEMBL7707821 0.76 AKT1 (0.48) STAT5BHSD11B1CTSLCTSSCTSB
SCHEMBL1010216 0.75 MEP1A (0.50) ABCB1CTSLCTSSPTGESCTSB
SCHEMBL12550044 0.75 STAT5B (0.49) STAT5BTAS2R14HSD11B1NR1H3PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144890-A1 METHOD FOR PREPARING HALOGENATED AMINES Wyeth (US) 2010-01-20 EP disclosed
WO-2008098103-A1 METHOD FOR PREPARING HALOGENATED AMINES WYETH (US) 2008-08-14 WO disclosed
US-20080188659-A1 Method for Preparing Halogenated Amines WYETH (US) 2008-08-07 US disclosed
US-20080188659-A1 Method for Preparing Halogenated Amines WYETH (US) 2008-08-07 US disclosed
US-20080188659-A1 Method for Preparing Halogenated Amines WYETH (US) 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188659-A1 Method for Preparing Halogenated Amines PNMT, ABL1, INMT STAT5B 3704/4885TAS2R14 3551/4885HSD11B1 2350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.