SCHEMBL3635480

SCHEMBL3635480

NC(=O)c1cccc2nc(-c3ccc(N4CCC(N)C4)cc3)[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.56
PRKD3 O94806 1/20 0.56
MAP4K4 O95819 1/20 0.56
PIM1 P11309 1/20 0.56
CLK2 P49760 1/20 0.56
MAP4K2 Q12851 1/20 0.56
CAMK2D Q13557 1/20 0.56
DYRK1A Q13627 1/20 0.56
PIM3 Q86V86 1/20 0.56
PRKD2 Q9BZL6 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56
STK17A Q9UEE5 1/20 0.56
MAP4K5 Q9Y4K4 1/20 0.56
AURKA O14965 1/20 0.45
PARP1 P09874 12/20 0.44
PARP2 Q9UGN5 9/20 0.44
CHEK2 O96017 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635473 0.83 AURKB (0.75) AURKBPRKD3MAP4K4PIM1CLK2
SCHEMBL3527499 0.83 AURKB (0.45) AURKBAURKAPARP1PARP2CHEK2
SCHEMBL3580358 0.83 PARP1 (0.53) AURKBPIM1PIM3AURKAPARP1
SCHEMBL3587289 0.82 AURKA (0.56) AURKBAURKAPARP1PARP2CHEK2
SCHEMBL3584716 0.81 AURKB (0.47) AURKBAURKAPARP1PARP2CHEK2
SCHEMBL3582373 0.79 PARP1 (0.49) AURKBPIM1PIM3AURKAPARP1
SCHEMBL3582282 0.79 AURKB (0.61) AURKBAURKAPARP1CHEK2
SCHEMBL3576982 0.79 AURKA (0.52) AURKBAURKAPARP1PARP2CHEK2
SCHEMBL3580122 0.79 AURKB (0.56) AURKBAURKAPARP1CHEK2
SCHEMBL3577227 0.78 AURKA (0.53) AURKBAURKAPARP1PARP2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed