SCHEMBL363587

SCHEMBL363587

Cc1cc(/C(CC(c2ccc(C(=O)NCCS(C)(=O)=O)cc2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.38
EPHX2 P34913 6/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
GPBAR1 Q8TDU6 4/20 0.34
PPARD Q03181 1/20 0.33
MAPK14 Q16539 1/20 0.33
GCG P01275 1/20 0.33
TP53 P04637 1/20 0.32
MDM2 Q00987 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363112 0.93 GPBAR1 (0.36) GCGREPHX2ALDH1A1POLBGPBAR1
SCHEMBL362797 0.91 GCGR (0.39) GCGREPHX2S1PR1S1PR3ALDH1A1
SCHEMBL363032 0.86 GPBAR1 (0.45) EPHX2POLBGPBAR1BRD4
SCHEMBL363811 0.85 S1PR1 (0.36) GCGREPHX2S1PR1S1PR3ALDH1A1
SCHEMBL362795 0.83 GPBAR1 (0.36) GCGREPHX2ALDH1A1POLBGPBAR1
SCHEMBL361680 0.83 GPBAR1 (0.47) GCGRS1PR1S1PR3POLBGPBAR1
SCHEMBL1390150 0.83 EPHX2 (0.35) GCGREPHX2S1PR1S1PR3GPBAR1
SCHEMBL1390151 0.83 EPHX2 (0.35) GCGREPHX2S1PR1S1PR3GPBAR1
SCHEMBL363696 0.82 BRD4 (0.36) GCGRS1PR1S1PR3ALDH1A1BRD4
SCHEMBL363248 0.80 GPBAR1 (0.41) S1PR1S1PR3GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed