SCHEMBL362797

SCHEMBL362797

Cc1cc(/C(CC(c2ccc(C(=O)NCCO)cc2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.39
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 2/20 0.38
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
EPHX2 P34913 2/20 0.36
GCG P01275 2/20 0.36
GPBAR1 Q8TDU6 3/20 0.35
BRD4 O60885 1/20 0.34
SLC6A3 Q01959 1/20 0.33
ANPEP P15144 1/20 0.33
SNCA P37840 2/20 0.33
S1PR2 O95136 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362795 0.93 GPBAR1 (0.36) GCGRALDH1A1POLBEPHX2GCG
SCHEMBL363696 0.91 BRD4 (0.36) GCGRS1PR1S1PR3ALDH1A1BRD4
SCHEMBL363587 0.91 GCGR (0.38) GCGRS1PR1S1PR3ALDH1A1POLB
SCHEMBL363811 0.90 S1PR1 (0.36) GCGRS1PR1S1PR3ALDH1A1POLB
SCHEMBL361680 0.86 GPBAR1 (0.47) GCGRS1PR1S1PR3POLBGPBAR1
SCHEMBL364032 0.85 GPBAR1 (0.47) ALDH1A1POLBEPHX2GPBAR1BRD4
SCHEMBL363638 0.85 GPBAR1 (0.41) S1PR1S1PR3GPBAR1
SCHEMBL363277 0.85 GPBAR1 (0.41) S1PR1S1PR3GPBAR1
SCHEMBL363248 0.85 GPBAR1 (0.41) S1PR1S1PR3GPBAR1
SCHEMBL363112 0.83 GPBAR1 (0.36) GCGRALDH1A1POLBEPHX2GCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed