SCHEMBL363696

SCHEMBL363696

Cc1cc(/C(CC(c2cccc(C(=O)NCCO)c2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
SNCA P37840 5/20 0.34
GPR52 Q9Y2T5 2/20 0.34
PNP P00491 1/20 0.34
GCGR P47871 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HAT1 O14929 3/20 0.33
EP300 Q09472 3/20 0.33
GPR139 Q6DWJ6 2/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362797 0.91 GCGR (0.39) BRD4S1PR1S1PR3SNCAGCGR
SCHEMBL362423 0.85 BRD4 (0.35) BRD4PNPCYP1A2CYP2D6CYP2C9
SCHEMBL362795 0.84 GPBAR1 (0.36) BRD4SNCAGCGRMEN1KMT2A
SCHEMBL363191 0.83 ALDH1A1 (0.38) BRD4S1PR1S1PR3PNPMEN1
SCHEMBL363587 0.82 GCGR (0.38) BRD4S1PR1S1PR3GCGRALDH1A1
SCHEMBL368824 0.82 CREBBP (0.35) BRD4SNCAGPR52MEN1KMT2A
SCHEMBL368825 0.82 CREBBP (0.35) BRD4SNCAGPR52MEN1KMT2A
SCHEMBL368826 0.82 CREBBP (0.35) BRD4SNCAGPR52MEN1KMT2A
SCHEMBL363811 0.81 S1PR1 (0.36) BRD4S1PR1S1PR3GCGRMEN1
SCHEMBL361680 0.79 GPBAR1 (0.47) BRD4S1PR1S1PR3GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed