SCHEMBL363687

SCHEMBL363687

C/C(=N/O)C(c1ccccc1)(c1ccc(Br)cc1)c1cc(Cl)nc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
NFKB1 P19838 1/20 0.31
CYP2C19 P33261 1/20 0.31
CASP3 P42574 1/20 0.31
NFKB2 Q00653 1/20 0.31
KMT2A Q03164 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
MCL1 Q07820 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363274 0.92 NPC1 (0.35) POLBNPC1RAB9AMEN1KMT2A
SCHEMBL365534 0.92 NPC1 (0.35) POLBNPC1RAB9AMEN1KMT2A
SCHEMBL364627 0.92 NPC1 (0.35) POLBNPC1RAB9AMEN1KMT2A
SCHEMBL364097 0.86 TRPA1 (0.35) POLB
SCHEMBL361971 0.83 NR1H2 (0.37) NPC1RAB9ANR1H2NR1H3MEN1
SCHEMBL3523097 0.75 KCNN4 (0.43) CYP1A2CYP3A4CYP2C19KMT2AALDH1A1
SCHEMBL3523100 0.75 KCNN4 (0.43) CYP1A2CYP3A4CYP2C19KMT2AALDH1A1
SCHEMBL364200 0.75 SMN1; SMN2 (0.34) POLBNPC1RAB9AMEN1CYP1A2
SCHEMBL365185 0.74 KIF11 (0.30)
SCHEMBL11403225 0.73 POLB (0.50) POLBNPC1RAB9AMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed