SCHEMBL361971

SCHEMBL361971

CC(=O)C(c1ccccc1)(c1ccc(Br)cc1)c1cc(Cl)nc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
KCNN4 O15554 4/20 0.36
TBXA2R P21731 2/20 0.36
PDE2A O00408 1/20 0.36
KIF11 P52732 1/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
HTT P42858 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
NFKB1 P19838 1/20 0.35
CYP2C19 P33261 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SENP7 Q9BQF6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363897 0.85 AR (0.36) NR1H2NR1H3KCNN4KIF11MEN1
SCHEMBL363687 0.83 POLB (0.36) NR1H2NR1H3TBXA2RPDE2AMEN1
SCHEMBL10538155 0.74 KIF11 (0.46) KCNN4KIF11MEN1KMT2ACYP1A2
SCHEMBL3523419 0.74 KCNN4 (0.58) KCNN4KMT2ACYP1A2CYP3A4CYP2C19
SCHEMBL364627 0.73 NPC1 (0.35) KCNN4MEN1KMT2ANPC1RAB9A
SCHEMBL365534 0.73 NPC1 (0.35) KCNN4MEN1KMT2ANPC1RAB9A
SCHEMBL363274 0.73 NPC1 (0.35) KCNN4MEN1KMT2ANPC1RAB9A
SCHEMBL11563715 0.70 HDAC3 (0.53) KIF11MEN1KMT2ANPC1CYP1A2
SCHEMBL364097 0.69 TRPA1 (0.35)
SCHEMBL365185 0.68 KIF11 (0.30) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed