SCHEMBL3646540

SCHEMBL3646540

Cc1ccc(S(=O)(=O)c2sc(C=O)cc2-c2cccnc2F)cn1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.36
PIP4K2A P48426 1/20 0.35
PIP4K2C Q8TBX8 1/20 0.35
CYP2A6 P11509 1/20 0.35
NAMPT P43490 4/20 0.33
KIT P10721 1/20 0.33
COMT P21964 1/20 0.32
PTGS1 P23219 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
PAX8 Q06710 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651198 0.88 KMT2A (0.38) PIP4K2APIP4K2CCYP2A6NAMPT
SCHEMBL3649066 0.87 FEN1 (0.39) CYP2A6
SCHEMBL3655764 0.85 CYP2A6 (0.39) PIP4K2APIP4K2CCYP2A6
SCHEMBL3691530 0.83 NAMPT (0.35) PIP4K2APIP4K2CCYP2A6NAMPT
SCHEMBL3654418 0.83 PIP4K2A (0.39) PTGS2PIP4K2APIP4K2CCYP2A6NAMPT
Fumaric Acid SCHEMBL4135457 0.76 NAMPT (0.37) PTGS2PIP4K2APIP4K2CCYP2A6NAMPT
Fumaric Acid SCHEMBL4135452 0.76 NAMPT (0.37) PTGS2PIP4K2APIP4K2CCYP2A6NAMPT
SCHEMBL3700772 0.76 CYP2A6 (0.39) PIP4K2APIP4K2CCYP2A6CA1CA2
SCHEMBL3655995 0.75 NFE2L2 (0.41) PIP4K2APIP4K2CCYP2A6
SCHEMBL3645616 0.74 CYP2A6 (0.37) CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-B1 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2014-12-31 EP disclosed
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
US-20090156642-A1 5-Membered heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156642-A1 5-Membered heterocyclic compound CEL, PGA5, COG5 PTGS2 269/4885PIP4K2A 1181/4885PIP4K2C 844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.