SCHEMBL3700772

SCHEMBL3700772

O=Cc1cc(-c2cccnc2F)c(S(=O)(=O)n2cccc2)s1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.39
PIP4K2A P48426 1/20 0.32
PIP4K2C Q8TBX8 1/20 0.32
ERN1 O75460 1/20 0.31
CYP2C19 P33261 1/20 0.30
GRIA2 P42262 1/20 0.30
DHODH Q02127 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL3695553 0.83 CYP2A6 (0.32) CYP2A6
SCHEMBL3655764 0.81 CYP2A6 (0.39) CYP2A6PIP4K2APIP4K2CDHODH
SCHEMBL3649066 0.78 FEN1 (0.39) CYP2A6CYP2C19
SCHEMBL3705487 0.77 CTSD (0.31) CYP2C19GRIA2CA1CA2
SCHEMBL2841100 0.76 CYP2A6 (0.50) CYP2A6PIP4K2APIP4K2CERN1CYP2C19
SCHEMBL3646540 0.76 PTGS2 (0.36) CYP2A6PIP4K2APIP4K2CCA1CA2
SCHEMBL3654418 0.76 PIP4K2A (0.39) CYP2A6PIP4K2APIP4K2C
SCHEMBL3691530 0.74 NAMPT (0.35) CYP2A6PIP4K2APIP4K2CERN1
Fumaric Acid SCHEMBL4132147 0.74 CYP2A6 (0.35) CYP2A6PIP4K2APIP4K2C
SCHEMBL3655995 0.73 NFE2L2 (0.41) CYP2A6PIP4K2APIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-B1 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2014-12-31 EP disclosed
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
US-20090156642-A1 5-Membered heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156642-A1 5-Membered heterocyclic compound CEL, PGA5, COG5 CYP2A6 443/4885PIP4K2A 1181/4885PIP4K2C 844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.