SCHEMBL3650693

SCHEMBL3650693

CN(Cc1cc(Sc2cccnc2)c(Br)s1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.36
HTR2C P28335 3/20 0.36
SLC6A4 P31645 3/20 0.36
RIPK1 Q13546 1/20 0.34
GLS O94925 2/20 0.34
SOS1 Q07889 1/20 0.32
RAB9A P51151 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CG P48736 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNA1B Q00975 1/20 0.31
CACNA1C Q13936 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
SSTR4 P31391 1/20 0.31
NAMPT P43490 2/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2A6 P11509 1/20 0.30
CYP2C19 P33261 1/20 0.30
MGLL Q99685 1/20 0.30
NR1D1 P20393 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132076 0.86 LMNA (0.37) CLK1RIPK1RAB9APIK3CAPIK3CG
SCHEMBL4118148 0.83 HTR2C (0.38) CLK1HTR2CSLC6A4RIPK1GLS
SCHEMBL3650699 0.79 NR1D1 (0.32) RIPK1RAB9APIK3CAPIK3CGNR1D1
SCHEMBL4137557 0.79 RIPK1 (0.36) CLK1HTR2CSLC6A4RIPK1GLS
SCHEMBL3649650 0.78 NAMPT (0.36) CLK1HTR2CSLC6A4RIPK1GLS
SCHEMBL3652849 0.73 HTR2C (0.41) HTR2CSLC6A4GLSSOS1CACNA1G
SCHEMBL3649821 0.73 SSTR4 (0.38) HTR2CSLC6A4GLSSOS1CACNA1G
SCHEMBL3650696 0.72 PIK3CA (0.35) RAB9APIK3CAPIK3CG
SCHEMBL5890773 0.71 RIPK1 (0.63) CLK1HTR2CSLC6A4RIPK1GLS
SCHEMBL4132086 0.71 SMN1; SMN2 (0.37) RAB9APIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed