SCHEMBL3650837

SCHEMBL3650837

CCCc1nc2nccc([N+](=O)[O-])c2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
ADORA3 P0DMS8 2/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
NOS2 P35228 5/20 0.38
NOS1 P29475 4/20 0.38
NOS3 P29474 3/20 0.38
PI4KA P42356 1/20 0.38
PI4K2B Q8TCG2 1/20 0.38
PI4K2A Q9BTU6 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
PIM3 Q86V86 1/20 0.38
GAA P10253 1/20 0.37
CYP3A4 P08684 3/20 0.36
CYP1A2 P05177 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9406926 0.78 ADORA1 (0.43) KDM4EADORA3ADORA2AADORA1NOS2
SCHEMBL7378689 0.76 NOS2 (0.59) ADORA3ADORA2AADORA1NOS2NOS1
SCHEMBL3964555 0.75 ADORA1 (0.43) KDM4EADORA3ADORA2AADORA1NOS2
SCHEMBL9406899 0.72 ADORA1 (0.42) KDM4EADORA3ADORA2AADORA1NOS2
SCHEMBL1892570 0.70 KDM4E (0.52) KDM4EADORA3NOS2NOS1GAA
SCHEMBL8561715 0.69 ADORA1 (0.41) ADORA3ADORA2AADORA1NOS2NOS1
SCHEMBL9041424 0.68 NOS1 (0.56) ADORA1NOS2NOS1NOS3PI4KA
SCHEMBL9648738 0.67 PI4KA (0.57) ADORA1NOS2NOS1NOS3PI4KA
SCHEMBL3507346 0.66 ALDH1A1 (0.44) KDM4ENOS2NOS1NOS3CYP3A4
SCHEMBL9406720 0.66 PI4KA (0.56) NOS2NOS1NOS3PI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185557-A2 PERHARIDINES AS CDK INHIBITORS Centre National De La Recherche Scientifique (FR) 2010-05-19 EP disclosed
WO-2009034475-A2 PERHARIDINES AS CDK INHIBITORS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2009-03-19 WO disclosed