SCHEMBL365148

SCHEMBL365148

COc1ccc(C(C(C)=O)(c2ccc(Br)cc2)c2ccccc2Cl)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
GPR183 P32249 3/20 0.38
RAB9A P51151 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
HTT P42858 2/20 0.37
PKM P14618 1/20 0.37
XBP1 P17861 1/20 0.37
MAPK1 P28482 1/20 0.37
AGTR1 P30556 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 3/20 0.36
POLB P06746 2/20 0.36
TSHR P16473 1/20 0.35
LIPE Q05469 1/20 0.35
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363964 0.87 GPR183 (0.38) SMN1; SMN2GPR183RAB9AALDH1A1MAPT
SCHEMBL14894794 0.87 GPR183 (0.38) SMN1; SMN2GPR183RAB9AALDH1A1MAPT
SCHEMBL363152 0.79 KCNN4 (0.45) SMN1; SMN2RAB9AALDH1A1MAPTHTT
SCHEMBL363254 0.75 TDO2 (0.36) SMN1; SMN2GPR183RAB9AALDH1A1MAPT
SCHEMBL364183 0.74 GPR183 (0.34) SMN1; SMN2GPR183RAB9AALDH1A1MAPT
SCHEMBL13427579 0.72 KCNN4 (0.48) SMN1; SMN2RAB9AALDH1A1MAPTHTT
SCHEMBL364659 0.72 KCNK3 (0.33) RAB9AALDH1A1MAPTPKMNPSR1
SCHEMBL14965127 0.71 KMT2A (0.38) SMN1; SMN2RAB9AALDH1A1MAPTNPSR1
SCHEMBL14965530 0.67 RAB9A (0.37) RAB9AMAPTMAPK1KMT2APOLB
SCHEMBL14965778 0.67 RAB9A (0.37) RAB9AMAPTMAPK1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed