SCHEMBL3652103

SCHEMBL3652103

COc1cccc(S(=O)(=O)c2sc(CN(CC(C)(C)C)C(=O)O)cc2-c2ccccc2F)c1.COc1cccc(S(=O)(=O)c2sc(CN(CC(C)(C)C)C(=O)O)cc2Br)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 1/20 0.36
TAS2R14 Q9NYV8 3/20 0.35
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
MEP1B Q16820 1/20 0.33
CHRM5 P08912 1/20 0.33
NFE2L2 Q16236 2/20 0.33
KEAP1 Q14145 1/20 0.33
PGR P06401 1/20 0.33
LPAR1 Q92633 1/20 0.33
LPAR5 Q9H1C0 1/20 0.33
HSD17B2 P37059 1/20 0.32
HSD11B1 P28845 1/20 0.32
LMNA P02545 3/20 0.32
ALDH1A1 P00352 2/20 0.32
POLB P06746 2/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651797 0.90 TAS2R14 (0.39) TAS2R14ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3649518 0.85 NFE2L2 (0.38) TAS2R14ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3652101 0.84 KAT6A (0.36) KAT6ATAS2R14ABCC9ABCC8KCNJ11
SCHEMBL3655896 0.82 KAT6A (0.42) KAT6ATAS2R14MEP1BCHRM5NFE2L2
SCHEMBL4029601 0.81 ABCC9 (0.36) TAS2R14ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3654647 0.81 CNR2 (0.35) HSD11B1LMNAALDH1A1HTTNPSR1
Carbamic Acid SCHEMBL3651238 0.78 CA12 (0.33) HSD11B1LMNAALDH1A1HTTNPSR1
SCHEMBL4131734 0.77 TAS2R14 (0.42) TAS2R14MEP1BCHRM5NFE2L2KEAP1
SCHEMBL3647498 0.76 C1S (0.33) KAT6A
SCHEMBL3646770 0.75 LMNA (0.30) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed