SCHEMBL365474

SCHEMBL365474

CS(=O)(=O)NC(=O)c1ccc(OCc2cccc(Cl)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.67
MAOA P21397 3/20 0.67
RXRA P19793 1/20 0.64
RXRB P28702 1/20 0.64
RXRG P48443 1/20 0.64
MRGPRX4 Q96LA9 3/20 0.55
ALOX5 P09917 1/20 0.55
BCL2L1 Q07817 1/20 0.54
MCL1 Q07820 1/20 0.54
NR4A2 P43354 1/20 0.53
ADAMTS4 O75173 1/20 0.52
MMP13 P45452 1/20 0.52
CYP4F2 P78329 1/20 0.52
CYP4A11 Q02928 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367348 0.89 BCL2L1 (0.57) MAOBMAOARXRARXRBRXRG
SCHEMBL365115 0.88 RXRA (0.64) MAOBMAOARXRARXRBRXRG
SCHEMBL16239839 0.85 MAOB (0.67) MAOBMAOAMRGPRX4ADAMTS4MMP13
SCHEMBL366713 0.85 RAB9A (0.57) MAOBMRGPRX4MMP13CYP4F2CYP4A11
SCHEMBL366081 0.85 MAOA (0.63) MAOBMAOABCL2L1MCL1NR4A2
SCHEMBL365210 0.85 MAOA (0.63) MAOBMAOABCL2L1MCL1NR4A2
SCHEMBL365173 0.84 MAOB (0.61) MAOBBCL2L1MCL1NR4A2
SCHEMBL10203178 0.84 SCN9A (0.66) MAOBMAOAMRGPRX4BCL2L1MCL1
Diethylamine SCHEMBL16239962 0.83 RXRA (0.58) MAOBMAOARXRARXRBRXRG
SCHEMBL363886 0.82 MAOB (0.69) MAOBMRGPRX4NR4A2ADAMTS4MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A MAOB 3660/4885MAOA 3705/4885RXRA 1658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.