SCHEMBL3658764

SCHEMBL3658764

COC(=O)c1ccc(C(CO)C(c2ccnc(C(=O)OC)c2)C(F)(F)F)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
PDK1 Q15118 2/20 0.37
PDK2 Q15119 2/20 0.37
PDK3 Q15120 2/20 0.37
PDK4 Q16654 2/20 0.37
CFTR P13569 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
MAPK1 P28482 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
AR P10275 1/20 0.34
KDM4E B2RXH2 1/20 0.33
KDM6B O15054 1/20 0.33
KDM5C P41229 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
ANO1 Q5XXA6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1414694 0.82 ALDH1A1 (0.38) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL3658227 0.81 MDM4 (0.38) PDK2MRGPRX4
SCHEMBL3658899 0.80 NR1H4 (0.37) PDK2MRGPRX4SMN1; SMN2RAB9ANPC1
SCHEMBL3803786 0.78 MRGPRX4 (0.37) ALDH1A1MRGPRX4SMN1; SMN2KDM4EKDM6B
SCHEMBL837022 0.73 PDK1 (0.43) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL3652084 0.71 P2RX7 (0.33) ALDH1A1SMN1; SMN2KDM4ERAB9ANPC1
SCHEMBL29878775 0.70 ALDH1A1 (0.43) ALDH1A1CFTRMAPK1CYP1A2CYP2C19
SCHEMBL3656229 0.69 ALDH1A1 (0.38) ALDH1A1MRGPRX4ARANO1NOTUM
SCHEMBL3659897 0.68 NR3C2 (0.37) ALDH1A1MRGPRX4SMN1; SMN2CYP1A2TSHR
SCHEMBL3660073 0.67 MAPT (0.32) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed