Quinupramine

Quinupramine

SCHEMBL366044

c1ccc2c(c1)CCc1ccccc1N2[C@@H]1CN2CCC1CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 1.00
CHRM1 P11229 3/20 1.00
HTR1A P08908 1/20 1.00
ADRA2A P08913 1/20 1.00
DRD1 P21728 1/20 1.00
SLC6A2 P23975 1/20 1.00
SLC6A4 P31645 1/20 1.00
ADRA1A P35348 1/20 1.00
OPRM1 P35372 1/20 1.00
DRD3 P35462 1/20 1.00
SLC6A3 Q01959 1/20 1.00
KCNH2 Q12809 1/20 1.00
CHRM3 P20309 2/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinupramine SCHEMBL29985275 1.00 CHRM2 (1.00) CHRM2CHRM1HTR1AADRA2ADRD1
Quinupramine SCHEMBL49100 1.00 CHRM2 (1.00) CHRM2CHRM1HTR1AADRA2ADRD1
Quinupramine SCHEMBL13280380 0.82 SLC6A4 (0.67) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL13471233 0.80 CHRM2 (0.66) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL13471238 0.80 ADRA2A (0.66) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL20216589 0.80 CHRM2 (0.66) CHRM2CHRM1HTR1AADRA2ADRD1
Amineptine SCHEMBL28280844 0.74 SLC6A3 (0.65) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL7281251 0.71 CHRM2 (0.55) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL7290543 0.71 CHRM2 (0.55) CHRM2CHRM1HTR1AADRA2ADRD1
SCHEMBL24903369 0.68 SLC18A3 (0.53) CHRM2CHRM1HTR1AADRA2ADRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 310 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117597126-A Pharmaceutical composition for preventing or treating cancer comprising CDK4/6 inhibitor and tricyclic antidepressant 国立癌症中心 2024-02-23 CN claimed
WO-2023282544-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT 국립암센터 2023-01-12 WO claimed
EP-2729136-A1 DRUG COMBINATIONS AND USES IN TREATING A COUGHING CONDITION Biocopea Limited (GB) 2014-05-14 EP claimed
WO-2013004999-A1 DRUG COMBINATIONS AND USES IN TREATING A COUGHING CONDITION BIOCOPEA LIMITED (GB) 2013-01-10 WO claimed
CN-102595894-A Compounds that treat malaria and prevent malaria transmission USA AS REPRESENTED BY THE SECRETARY DEPT OF HEALTH AND HUMAN SERVICES 2012-07-18 CN claimed
CN-101132777-A Pharmaceutical compositions for sleep disorders COLLEGIUM PHARMACEUTICAL INC (US) 2008-02-27 CN claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-12564596-B2 Agents and methods for modulating pathogen activity GRIFFITH UNIVERSITY (AU) 2026-03-03 US disclosed
US-12527799-B2 Treatment of autism spectrum disorders, obsessive-compulsive disorder and anxiety disorders RUGEN HOLDINGS (CAYMAN) LIMITED (KY) 2026-01-20 US disclosed
US-20250241910-A1 COMBINATION THERAPY FOR THE TREATMENT OF PSYCHIATRIC DISORDER GSKB Pharmaceuticals, LLC 2025-07-31 US disclosed
US-20250152601-A1 Compositions and Methods for the Treatment of Sexual Dysfunctions THE JONATHAN HURT LIVING TRUST (US) 2025-05-15 US disclosed
US-20240350483-A1 COMBINATION THERAPY FOR THE TREATMENT OF PSYCHIATRIC DISORDER GSKB Pharmaceuticals, LLC 2024-10-24 US disclosed
EP-0737066-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1996-10-16 EP disclosed
EP-0710106-A1 METHOD OF TREATING ADDICTIVE BEHAVIORS HITZIG, Pietr (US) 1996-05-08 EP disclosed
US-5502080-A Combined use of dopamine and serotonin agonists in the treatment of allergic disorders HITZIG PIETR (US) 1996-03-26 US disclosed
US-5446070-A Flexible, finite, bioadhesive, therapeutical agent in solid form NOVER PHARMACEUTICALS, INC. (US) 1995-08-29 US disclosed
WO-1995018603-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1995-07-13 WO disclosed
WO-1994021244-A1 METHOD OF TREATING ADDICTIVE BEHAVIORS HITZIG PIETR (US) 1994-09-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12564596-B2 Agents and methods for modulating pathogen activity C3AR1, HTR3A, CHRM3 CHRM2 18/4885CHRM1 12/4885HTR1A 26/4885
US-20240350483-A1 COMBINATION THERAPY FOR THE TREATMENT OF PSYCHIATRIC DISORDER SLC6A4, SLC6A2, SLC6A3 CHRM2 1532/4885CHRM1 2063/4885HTR1A 20/4885
US-12527799-B2 Treatment of autism spectrum disorders, obsessive-compulsive disorder and anxiety disorders GRIN2C, GRIN3A, GRIN1 CHRM2 805/4885CHRM1 404/4885HTR1A 45/4885
US-20250241910-A1 COMBINATION THERAPY FOR THE TREATMENT OF PSYCHIATRIC DISORDER SLC6A4, SLC6A2, SLC6A3 CHRM2 1532/4885CHRM1 2063/4885HTR1A 20/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.