SCHEMBL366076

SCHEMBL366076

COc1cc(O)cc2c1c(C(=O)O)c1ccccn12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
MAPT P10636 5/20 0.40
ATM Q13315 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KCNA3 P22001 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
IDO1 P14902 2/20 0.39
NPC1 O15118 2/20 0.39
GAA P10253 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365191 0.88 MKNK2 (0.40) MAPTATMMEN1KMT2AKCNA3
SCHEMBL365175 0.87 NPC1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL366558 0.85 NPC1 (0.42) CA12CA1CA2CA7CA9
SCHEMBL367749 0.84 NPC1 (0.41) CA12CA1CA2CA7CA9
SCHEMBL366033 0.82 NPC1 (0.40) CA12CA1CA2CA7CA9
SCHEMBL366019 0.81 STS (0.41) CA12CA1CA2CA7CA9
SCHEMBL367733 0.80 KMT2A (0.38) CA12CA1CA2CA7CA9
SCHEMBL365272 0.79 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL365105 0.78 ALDH1A1 (0.43) MAPTATMMEN1KMT2ANPC1
SCHEMBL365225 0.77 CA12 (0.35) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed