SCHEMBL366033

SCHEMBL366033

COc1cc(C(=O)N(C)C)cc2c1c(C(=O)O)c1ccccn12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
ATM Q13315 2/20 0.40
GAA P10253 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CYP19A1 P11511 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
ACLY P53396 2/20 0.38
ERN1 O75460 1/20 0.38
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366817 0.90 NPC1 (0.39) NPC1ATMGAARXFP1CYP19A1
SCHEMBL365175 0.89 NPC1 (0.43) NPC1ATMGAARXFP1KDM4E
SCHEMBL366558 0.87 NPC1 (0.42) NPC1ATMGAARXFP1KDM4E
SCHEMBL367749 0.86 NPC1 (0.41) NPC1ATMGAARXFP1KDM4E
SCHEMBL366789 0.84 IDO1 (0.38) KDM4EALDH1A1MAPTACLYERN1
SCHEMBL367733 0.82 KMT2A (0.38) NPC1ATMGAARXFP1KDM4E
SCHEMBL366076 0.82 CA12 (0.41) NPC1ATMGAARXFP1KDM4E
SCHEMBL365272 0.81 CA12 (0.42) NPC1ATMGAARXFP1KDM4E
SCHEMBL367204 0.79 RORC (0.43) GAAKDM4EALDH1A1MAPTFNTA
SCHEMBL367176 0.79 HTR6 (0.38) KDM4EALDH1A1MAPTIDO1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed