SCHEMBL367733

SCHEMBL367733

COc1cc(OC(=O)N(C)C)cc2c1c(C(=O)O)c1ccccn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.38
NCEH1 Q6PIU2 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 2/20 0.35
NPC1 O15118 2/20 0.35
GAA P10253 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
MEN1 O00255 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
IDO1 P14902 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365489 0.90 KMT2A (0.36) KMT2AALDH1A1PKMNCEH1RAB9A
SCHEMBL365212 0.86 KMT2A (0.39) KMT2AALDH1A1PKMNCEH1RAB9A
SCHEMBL365188 0.85 CYP11B1 (0.39) KMT2AALDH1A1PKMLMNA
SCHEMBL366033 0.82 NPC1 (0.40) ALDH1A1ATMNPC1GAARXFP1
SCHEMBL365768 0.82 ALOX5 (0.38) KMT2AALDH1A1PKMRAB9ANPC1
SCHEMBL366019 0.81 STS (0.41) KMT2AALDH1A1ATMNPC1GAA
SCHEMBL365592 0.80 MRGPRX4 (0.39) KMT2AALDH1A1PKMRAB9ANPC1
SCHEMBL366850 0.80 MAPT (0.37) KMT2AALDH1A1RXFP1MEN1KDM4E
SCHEMBL366113 0.80 EPHX1 (0.49) KMT2ARAB9ANPC1GAAMEN1
SCHEMBL365175 0.80 NPC1 (0.43) ALDH1A1PKMATMNPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed