SCHEMBL366019

SCHEMBL366019

COc1cc(OS(N)(=O)=O)cc2c1c(C(=O)O)c1ccccn12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 6/20 0.41
IDO1 P14902 2/20 0.38
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
PTGS2 P35354 1/20 0.37
ATM Q13315 2/20 0.36
CA12 O43570 1/20 0.35
CA7 P43166 1/20 0.35
CA14 Q9ULX7 1/20 0.35
NPC1 O15118 2/20 0.35
GAA P10253 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
FABP4 P15090 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
MEN1 O00255 1/20 0.35
APAF1 O14727 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367759 0.91 STS (0.41) STSIDO1CA1CA2CA9
SCHEMBL365225 0.86 CA12 (0.35) IDO1CA1CA2CA9PTGS2
SCHEMBL366115 0.86 CA1 (0.41) STSIDO1CA1CA2CA9
SCHEMBL367733 0.81 KMT2A (0.38) IDO1CA1CA2CA9ATM
SCHEMBL365175 0.81 NPC1 (0.43) IDO1CA1CA2CA9PTGS2
SCHEMBL366076 0.81 CA12 (0.41) IDO1CA1CA2CA9PTGS2
SCHEMBL367749 0.80 NPC1 (0.41) CA1CA2CA9PTGS2ATM
SCHEMBL365105 0.79 ALDH1A1 (0.43) PTGS2ATMNPC1GAARXFP1
SCHEMBL366074 0.79 POLB (0.33) IDO1ATMNPC1GAARXFP1
SCHEMBL366558 0.79 NPC1 (0.42) IDO1CA1CA2CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed