SCHEMBL366128

SCHEMBL366128

COc1ccc(C(=O)[C@@H](N)CN2CCCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.64
LMNA P02545 4/20 0.64
SMN1; SMN2 Q16637 3/20 0.64
MITF O75030 2/20 0.64
HIF1A Q16665 1/20 0.64
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
SLC6A3 Q01959 1/20 0.54
POLB P06746 3/20 0.53
MAPT P10636 3/20 0.53
HTT P42858 2/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HPGD P15428 1/20 0.51
KDM4E B2RXH2 1/20 0.51
DRD3 P35462 2/20 0.50
DRD2 P14416 1/20 0.50
CHRM2 P08172 1/20 0.49
ADRA2B P18089 1/20 0.49
SIGMAR1 Q99720 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10854806 0.83 DRD3 (0.72) ALDH1A1LMNASMN1; SMN2MITFHIF1A
Hydrochloric Acid SCHEMBL10896084 0.82 ALDH1A1 (0.72) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL23094153 0.79 SMN1; SMN2 (1.00) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL6864368 0.79 ALDH1A1 (0.62) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL10851628 0.78 SMN1; SMN2 (0.97) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL28859465 0.77 CA1 (0.53) ALDH1A1LMNASMN1; SMN2HTTMEN1
Hydrochloric Acid SCHEMBL10851947 0.77 LMNA (0.95) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL28859493 0.76 KIF11 (0.56) ALDH1A1LMNASMN1; SMN2HTTMEN1
SCHEMBL13037583 0.75 ALPL (0.55) ALDH1A1LMNASMN1; SMN2MITFHIF1A
SCHEMBL10256789 0.74 SMN1; SMN2 (0.64) ALDH1A1LMNASMN1; SMN2MITFHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2198864-B1 Pharmaceutical compositions having an analgesic effect and containing 1-benzyl-1-hydroxy-2,3-diamino-propyl amines, 3-benzyl-3-hydroxy-2-amino propionic acid amides or related compounds ALLERGAN INC (US) 2012-03-14 EP disclosed