SCHEMBL366238

SCHEMBL366238

CC(=O)c1ccc2c(C(=O)CCCCN(C)C)c3ccccn3c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
PRNP P04156 1/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
CHRM1 P11229 1/20 0.44
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
TBXA2R P21731 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
ADRA1A P35348 1/20 0.44
OPRM1 P35372 1/20 0.44
DRD3 P35462 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KCNH2 Q12809 1/20 0.44
PLA2G2A P14555 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366185 0.92 CYP1A2 (0.42) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL365468 0.87 ALDH1A1 (0.39) CYP1A2PLA2G2AMAPTMEN1KMT2A
SCHEMBL367618 0.86 BAZ2B (0.38) HTR1AADRA2ADRD2DRD1SLC6A2
SCHEMBL366837 0.85 ALDH1A1 (0.40) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL364304 0.85 CHRM1 (0.38) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL366239 0.82 PLA2G2A (0.41) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL365487 0.82 POLR1A (0.40) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL366441 0.81 ALDH1A1 (0.43) CYP1A2LMNATP53MAPTMEN1
SCHEMBL366299 0.80 LMNA (0.38) CYP1A2CYP2D6TSHRLMNAPRNP
SCHEMBL364861 0.80 EGFR (0.51) CYP1A2CYP2D6LMNAKCNH2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed