SCHEMBL3665110

SCHEMBL3665110

CN(C)C(CCc1ccccc1)C1CCC(CC(CNC(=O)c2ccccc2O)Oc2ccccc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NLRP1 Q9C000 1/20 0.39
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
PNLIP P16233 2/20 0.34
ESRRG P62508 1/20 0.34
OPRM1 P35372 4/20 0.34
NAPEPLD Q6IQ20 1/20 0.34
P2RX7 Q99572 1/20 0.33
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3666093 0.84 OPRM1 (0.37) ALDH1A1HPGDTSHRHSD17B10MEN1
SCHEMBL3666492 0.80 P2RX7 (0.38) MAPTMEN1KMT2APNLIPOPRM1
SCHEMBL3666118 0.78 OPRL1 (0.38) MEN1KMT2AOPRM1P2RX7
SCHEMBL493639 0.74 MAPT (0.44) ALDH1A1MAPTMEN1KMT2ANAPEPLD
SCHEMBL493440 0.70 TSHR (0.48) ALDH1A1HPGDNPC1MAPTTSHR
SCHEMBL1327183 0.69 CHRNB2 (0.39) NPC1OPRM1KDM4ESMN1; SMN2L3MBTL1
SCHEMBL1328400 0.69 KMT2A (0.38) ALDH1A1HPGDTSHRHTTMEN1
SCHEMBL493155 0.68 SMN1; SMN2 (0.50) MAPTMEN1KMT2ANAPEPLDSMN1; SMN2
SCHEMBL2308766 0.67 KDM4E (0.42) ALDH1A1HPGDNPC1TSHRHSD17B10
SCHEMBL493056 0.67 SLC6A2 (0.37) OPRM1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP claimed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO claimed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP disclosed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO disclosed