SCHEMBL3666093

SCHEMBL3666093

CN(C)C(c1ccccc1)C1CCC(CC(CNC(=O)c2ccccc2O)Oc2ccccc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.37
P2RX7 Q99572 4/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 1/20 0.36
PNLIP P16233 2/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3666492 0.94 P2RX7 (0.38) OPRM1P2RX7KDM4EPNLIPMEN1
SCHEMBL3666118 0.92 OPRL1 (0.38) OPRM1P2RX7MEN1KMT2ATDP1
SCHEMBL3665110 0.84 ALDH1A1 (0.39) OPRM1P2RX7KDM4EALDH1A1HPGD
SCHEMBL2308766 0.79 KDM4E (0.42) OPRM1KDM4EALDH1A1LMNAHPGD
SCHEMBL2306855 0.74 HTR7 (0.45) P2RX7KDM4EALDH1A1HPGD
SCHEMBL1327800 0.72 HPGD (0.44) P2RX7ALDH1A1HPGDMEN1KMT2A
SCHEMBL493195 0.72 GAA (0.46) ALDH1A1HPGDTSHRMEN1KMT2A
SCHEMBL1327283 0.71 KCNA3 (0.50) OPRM1P2RX7KDM4EALDH1A1LMNA
SCHEMBL1326883 0.71 ALDH1A1 (0.44) OPRM1KDM4EALDH1A1TSHRMEN1
SCHEMBL1327964 0.71 NPC1 (0.50) P2RX7KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP claimed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO claimed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP disclosed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO disclosed