SCHEMBL366512

SCHEMBL366512

Cn1nccc1-c1cc(Cl)ccc1OCc1ccc(C(=O)NS(C)(=O)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 9/20 0.51
SCN9A Q15858 2/20 0.50
SCN5A Q14524 1/20 0.50
HTR2A P28223 9/20 0.47
HTR2C P28335 8/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diethylamine SCHEMBL16240132 0.96 PTGER1 (0.47) PTGER1SCN9ASCN5AHTR2AHTR2C
SCHEMBL16319570 0.85 SCN9A (0.51) SCN9ASCN5AHTR2AHTR2C
SCHEMBL16242182 0.80 SCN9A (0.58) SCN9AHTR2AHTR2C
SCHEMBL364759 0.79 MRGPRX4 (0.64) SCN9ASCN5A
SCHEMBL16319802 0.79 SCN9A (0.63) SCN9A
SCHEMBL365276 0.78 BCL2L1 (0.47) SCN9ASCN5A
SCHEMBL16240302 0.78 MRGPRX4 (0.61) SCN9ASCN5A
SCHEMBL364527 0.75 SCN9A (0.63) SCN9ASCN5A
Diethylamine SCHEMBL16239865 0.75 MRGPRX4 (0.58) SCN9ASCN5A
Diethylamine SCHEMBL16239843 0.74 CYP1A2 (0.46) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A PTGER1 372/4885SCN9A 16/4885SCN5A 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.