SCHEMBL3666428

SCHEMBL3666428

Fc1cccc(C2CNCC[N]2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
NOS3 P29474 1/20 0.40
NISCH Q9Y2I1 1/20 0.37
HTR6 P50406 7/20 0.37
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.36
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CA1 P00915 1/20 0.35
IDO1 P14902 1/20 0.35
HTR7 P34969 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240396 0.81 HTR2C (0.50) NISCHHTR2CHTR2BHTR2ANPC1
SCHEMBL1254610 0.81 SLC6A3 (0.44) TAAR1HTR2CHTR2BHTR2A
SCHEMBL1255265 0.80 HTR1A (0.55) HTR2CHTR2BHTR2A
SCHEMBL1616732 0.80 KDM1A (0.38) NOS3
SCHEMBL571789 0.79 SLC18A3 (0.41) TAAR1NISCHNFKB1
SCHEMBL4374233 0.77 CHRNB2 (0.40) HTR6HTR2CHTR2BHTR2A
SCHEMBL2218295 0.77 HTR2C (0.54) NISCHHTR2CHTR2BHTR2ANPC1
SCHEMBL8658279 0.75
SCHEMBL3151536 0.75 TAAR1 (0.47) TAAR1NOS3HTR2CHTR2BHTR2A
SCHEMBL7289047 0.74 MAOA (0.40) HTR2CSMN1; SMN2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150532-A1 PIPERAZINE COMPOUNDS FOR THE INHIBITION OF HAEMATOPOIETIC PROSTAGLANDIN D SYNTHASE Evotec AG (DE) 2010-02-10 EP disclosed
WO-2008122787-A1 PIPERAZINE COMPOUNDS FOR THE INHIBITION OF HAEMATOPOIETIC PROSTAGLANDIN D SYNTHASE EVOTEC AG (DE) 2008-10-16 WO disclosed