SCHEMBL366817

SCHEMBL366817

COc1cc(C(=O)N(C)C)cc2c1c(C(N)=O)c1ccccn12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CYP19A1 P11511 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
ERN1 O75460 1/20 0.37
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
RAB9A P51151 1/20 0.35
F10 P00742 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366033 0.90 NPC1 (0.40) NPC1GAAATMRXFP1CYP19A1
SCHEMBL367765 0.89 NPC1 (0.43) NPC1GAAATMRXFP1KDM4E
SCHEMBL365272 0.87 CA12 (0.42) NPC1GAAATMRXFP1KDM4E
SCHEMBL365020 0.87 BAZ2B (0.43) NPC1GAAATMRXFP1KDM4E
SCHEMBL364537 0.85 BAZ2B (0.38) CYP19A1KDM4EALDH1A1MAPTERN1
SCHEMBL367749 0.82 NPC1 (0.41) NPC1GAAATMRXFP1KDM4E
SCHEMBL365489 0.82 KMT2A (0.36) ALDH1A1RAB9A
SCHEMBL365191 0.82 MKNK2 (0.40) NPC1GAAATMRXFP1KDM4E
SCHEMBL365916 0.80 KDM4E (0.40) GAAKDM4EALDH1A1MAPTERN1
SCHEMBL365175 0.78 NPC1 (0.43) NPC1GAAATMRXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed