SCHEMBL3668817

SCHEMBL3668817

COc1ccc2nccc(C3(O)CCN(C(=O)O)CC3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP8B1 Q9UNU6 1/20 0.37
KCNH2 Q12809 6/20 0.37
SLC2A1 P11166 3/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
PKLR P30613 3/20 0.35
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1224264 0.86 MAP4K4 (0.42) CYP8B1
SCHEMBL1224605 0.80 SIGMAR1 (0.45) KCNH2SLC2A1PIK3CA
SCHEMBL14539419 0.78 KCNH2 (0.38) KCNH2SLC2A1
SCHEMBL1222813 0.77 KCNH2 (0.40) KCNH2SLC2A1
SCHEMBL21061155 0.72 PKLR (0.44) PKLR
SCHEMBL3662100 0.72 LMNA (0.43) KCNH2
SCHEMBL3960269 0.68 KCNH2 (0.41) KCNH2
SCHEMBL5309028 0.68 LMNA (0.43) KCNH2
SCHEMBL2790975 0.68 ALDH1A1 (0.40) KCNH2
Oxalic Acid SCHEMBL5255846 0.67 POLB (0.40) CYP8B1KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144910-A2 OXAZOLIDINONE ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2010-01-20 EP disclosed
WO-2008126034-A2 OXAZOLIDINONE ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2008-10-23 WO disclosed