SCHEMBL2790975

SCHEMBL2790975

COc1ccc(C2(O)CCN(C(=O)O)C2)cn1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.39
KCNH2 Q12809 3/20 0.39
NPY1R P25929 1/20 0.39
SLC6A4 P31645 1/20 0.39
NNMT P40261 1/20 0.38
CCR2 P41597 3/20 0.38
KDM4E B2RXH2 1/20 0.37
GRIN2B Q13224 1/20 0.37
SCN9A Q15858 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
GPR183 P32249 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3662100 0.92 LMNA (0.43) ALDH1A1LMNAKCNH2NPY1RSLC6A4
SCHEMBL23112352 0.89 NNMT (0.42) ALDH1A1LMNAKCNH2NNMTCCR2
SCHEMBL3469434 0.84 GPR119 (0.48)
SCHEMBL5468647 0.80 MAPT (0.47) ALDH1A1LMNAKCNH2CCR2CYP2D6
SCHEMBL3024794 0.79 GPR119 (0.53) ALDH1A1LMNACCR2
SCHEMBL23647652 0.79 NNMT (0.43) ALDH1A1LMNAKCNH2NPY1RSLC6A4
SCHEMBL29457438 0.78 GPR119 (0.47) CCR2MEN1KMT2A
SCHEMBL27210984 0.78 GPR119 (0.47) CCR2MEN1KMT2A
SCHEMBL5462315 0.78 GHSR (0.44) ALDH1A1LMNACYP2D6HPGDMEN1
SCHEMBL2264503 0.77 HDAC3 (0.48) GRIN2BSCN9ACYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010051245-A1 BENZIMIDAZOLE AND AZA-BENZIMIDAZOLE CARBOXAMIDES MERCK SHARP & DOHME CORP. (US) 2010-05-06 WO disclosed