SCHEMBL3670124

SCHEMBL3670124

Cc1c(Cl)cccc1NNC1=NCCN1.c1ccc(CNC2=NCCN2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 9/20 0.48
PTGIR P43119 1/20 0.47
ADRA2B P18089 5/20 0.45
ADRA2C P18825 5/20 0.45
ADRA2A P08913 4/20 0.45
ADRA1A P35348 4/20 0.45
HTR7 P34969 2/20 0.45
ADRA1D P25100 3/20 0.43
ADRA1B P35368 3/20 0.43
LMNA P02545 2/20 0.43
NISCH Q9Y2I1 2/20 0.43
MEN1 O00255 1/20 0.43
SLC22A1 O15245 1/20 0.43
SLC22A3 O75751 1/20 0.43
HTR1A P08908 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HRH2 P25021 1/20 0.43
CYP2C19 P33261 1/20 0.43
OPRK1 P41145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3169026 0.87 ADRA2A (0.55) PTGIRADRA2BADRA2CADRA2AADRA1A
SCHEMBL3169468 0.79 PTGIR (0.60) WDR5PTGIRADRA2BADRA2CADRA2A
SCHEMBL27797575 0.79 WDR5 (0.45) WDR5PTGIRADRA2BADRA2CADRA2A
SCHEMBL8148008 0.77 LMNA (0.52) WDR5PTGIRADRA2BADRA2CADRA2A
SCHEMBL11591507 0.76 ADRA2A (0.57) PTGIRADRA2BADRA2CADRA2AADRA1A
SCHEMBL29412295 0.75 ADRA2A (0.65) ADRA2BADRA2CADRA2AADRA1AHTR7
Hydrochloric Acid SCHEMBL11513827 0.75 ADRA2A (0.58) PTGIRADRA2BADRA2CADRA2AADRA1A
SCHEMBL11198769 0.74 ADRA2A (0.58) PTGIRADRA2BADRA2CADRA2AADRA1A
SCHEMBL11203702 0.74 ADRA2A (0.60) ADRA2BADRA2CADRA2AADRA1AHTR7
SCHEMBL10965126 0.72 ADRA2C (0.74) ADRA2BADRA2CADRA2AADRA1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173720-A2 2-IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. Hoffmann-Roche AG (CH) 2010-04-14 EP claimed
WO-2009003868-A2 2 -IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. HOFFMANN-LA ROCHE AG (CH) 2009-01-08 WO claimed