SCHEMBL3672155

SCHEMBL3672155

CCc1c(Br)ccc(N)c1N

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
AXL P30530 1/20 0.31
S100B P04271 1/20 0.31
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SKP2 Q13309 1/20 0.31
CD44 P16070 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB2 P47870 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8467859 0.84 NOS3 (0.33) NOS3NOS2AXLS100BALDH1A1
SCHEMBL7060663 0.80 NOS3 (0.37) NOS3NOS2S100BALDH1A1MEN1
SCHEMBL14994586 0.80 CYP3A4 (0.37) NOS3NOS2AXLS100BALDH1A1
SCHEMBL20475215 0.78 HTR1D (0.33) NOS3NOS2
SCHEMBL4513208 0.76 NOS3 (0.35) NOS3NOS2AXLS100BALDH1A1
SCHEMBL571458 0.74 POLB (0.40) NOS3NOS2ALDH1A1POLBMAPT
SCHEMBL982159 0.74 NOS2 (0.47) NOS3NOS2S100BALDH1A1POLB
SCHEMBL3669302 0.73 CYP3A4 (0.35) NOS3NOS2ALDH1A1CD44CYP3A4
SCHEMBL6204770 0.73 GABRA1 (0.39) NOS3NOS2ALDH1A1CD44GABRA1
SCHEMBL979815 0.73 ALDH1A1 (0.34) NOS3NOS2S100BALDH1A1CD44

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177604-A1 HETEROCYCLIC KINASE INHIBITORS Bristol-Myers Squibb Company (US) 2017-06-14 EP disclosed
WO-2016022312-A1 HETEROCYCLIC KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2016-02-11 WO disclosed
EP-1426392-B1 COMPOSITION FOR OPTICAL MATERIAL MITSUBISHI GAS CHEMICAL CO (JP) 2010-02-24 EP disclosed
US-6960640-B2 Composition for optical material MITSUBISHI GAS CHEMICAL CO., LTD. (JP) 2005-11-01 US disclosed
US-20040147708-A1 Composition for optical material MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2004-07-29 US disclosed
EP-1426392-A1 COMPOSITION FOR OPTICAL MATERIAL MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2004-06-09 EP disclosed