SCHEMBL367474

SCHEMBL367474

CCOC(=O)N1c2ccccc2C=CC1OCC.CCOC(=O)N1c2ccccc2C=CC1OCC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 1.00
LMNA P02545 2/20 1.00
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
P2RX4 Q99571 6/20 0.42
BCHE P06276 1/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPK1 P28482 2/20 0.41
TSHR P16473 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GAA P10253 1/20 0.41
P2RX1 P51575 3/20 0.38
P2RX3 P56373 3/20 0.38
P2RX7 Q99572 2/20 0.38
PTBP1 P26599 1/20 0.38
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL338 1.00 SMN1; SMN2 (1.00) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL29367804 1.00 SMN1; SMN2 (1.00) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL23705539 1.00 SMN1; SMN2 (1.00) SMN1; SMN2LMNAMEN1KMT2AP2RX4
Carbimide SCHEMBL10800076 0.95 SMN1; SMN2 (0.90) SMN1; SMN2LMNAMEN1KMT2AP2RX4
1,2-Dichloroethane SCHEMBL28697158 0.95 SMN1; SMN2 (0.90) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL8608444 0.93 SMN1; SMN2 (0.86) SMN1; SMN2LMNAMEN1KMT2AP2RX4
Dimethylformamide SCHEMBL7714545 0.92 SMN1; SMN2 (0.84) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL8063974 0.91 SMN1; SMN2 (0.82) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL8608446 0.91 SMN1; SMN2 (0.82) SMN1; SMN2LMNAMEN1KMT2AP2RX4
SCHEMBL9188247 0.90 SMN1; SMN2 (0.82) SMN1; SMN2LMNAMEN1KMT2AP2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 448 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486771-A Thiocarbonate-based hydrogen sulfide donor, and preparation method and application thereof 上海交通大学 2024-02-02 CN claimed
WO-2019200764-A1 IMPROVED CELLULOSE AND PREPARATION METHOD AND APPLICATION THEREFOR 东莞理工学院 2019-10-24 WO claimed
US-20240209001-A1 HETEROCYCLIC DERIVATIVES AS JANUS KINASE INHIBITORS Chiesi Farmaceutici S.p. A. (IT) 2024-06-27 US disclosed
US-20240197898-A1 SUBSTITUTED BENZO[5,6][1,4]DIAZEPINO[1,2-a]INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS IMMUNOGEN, INC. 2024-06-20 US disclosed
US-20240182464-A1 SELECTIVE BCL-XL PROTAC COMPOUNDS AND METHODS OF USE Les Laboratoirens Serviece (FR) 2024-06-06 US disclosed
EP-4376886-A2 METHODS OF TREATING CANCER Foghorn Therapeutics Inc. (US) 2024-06-05 EP disclosed
CN-107108507-B Process for preparing diaryl thiohydantoin compounds 阿拉贡药品公司 2024-05-28 CN disclosed
US-11981687-B2 Methods of preparing cytotoxic benzodiazepine derivatives IMMUNOGEN, INC. (US) 2024-05-14 US disclosed
CN-110637011-B Fanisole X receptor agonist and application thereof 奥加诺沃公司 2024-05-14 CN disclosed
CN-118043053-A Methods of treating cancer 福宏治疗公司 2024-05-14 CN disclosed
CN-110637015-B Fanisole X receptor agonist and application thereof 奥加诺沃公司 2024-04-02 CN disclosed
WO-1997006138-A1 4-MERCAPTOPYRROLIDINE DERIVATIVES AS FARNESYL TRANSFERASE INHIBITORS ZENECA LIMITED (GB) 1997-02-20 WO disclosed
EP-0694036-A1 HYDROXAMIC ACID DERIVATIVES BRITISH BIOTECH PHARM (GB) 1996-01-31 EP disclosed
WO-1994024140-A1 HYDROXAMIC ACID DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1994-10-27 WO disclosed
US-5324786-A Process for preparation of a solid phase system ORPEGEN MEDIZINISCHE-MOLEKULAR BIOLOGISCHE FORSCHUNGSGESELLSCHAFT MBH (DE) 1994-06-28 US disclosed
US-5214195-A ALLYL ESTERS AND THE USE THEREOF FOR THE BUILD-UP OF SOLID PHASE SYSTEMS FOR SOLID PHASE REACTIONS ORPEGEN MEDIZINISCH-MOLEKULAR BIOLOGISCHE FORSCHUNGSGESELLSCHAFT MBH (DE) 1993-05-25 US disclosed
EP-0415331-A2 Allyl esters and their application to the construction of solid phase systems for solid phase reactions Orpegen Medizinisch-Molekularbiologische Forschungsgesellschaft m.b.H. (DE) 1991-03-06 EP disclosed
EP-0298820-A1 Peptide derivatives and their therapeutic application INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1989-01-11 EP disclosed
US-4066831-A ANTIBIOTICS BRISTOL-MYERS COMPANY (US) 1978-01-03 US disclosed
US-4012383-A BACTERICIDES BRISTOL-MYERS COMPANY (US) 1977-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11981687-B2 Methods of preparing cytotoxic benzodiazepine derivatives GABRA3, GABRA5, GABRA6 SMN1; SMN2 2230/4885LMNA 945/4885MEN1 2163/4885
US-20240197898-A1 SUBSTITUTED BENZO[5,6][1,4]DIAZEPINO[1,2-a]INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS MKI67, GABBR1, GABBR2 SMN1; SMN2 3393/4885LMNA 2428/4885MEN1 1230/4885
US-20240182464-A1 SELECTIVE BCL-XL PROTAC COMPOUNDS AND METHODS OF USE CRBN, XIAP, BCL2L11 SMN1; SMN2 2309/4885LMNA 645/4885MEN1 3679/4885
US-20240209001-A1 HETEROCYCLIC DERIVATIVES AS JANUS KINASE INHIBITORS TYK2, JAK3, JAK1 SMN1; SMN2 4462/4885LMNA 4155/4885MEN1 4286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.