SCHEMBL5772791

SCHEMBL5772791

COc1cccc2c(CC(=O)N3CCC(NCc4ccc5cc(O)ccc5n4)CC3)ccnc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
ADORA2A P29274 3/20 0.36
MC4R P32245 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
SYK P43405 2/20 0.35
TACR1 P25103 3/20 0.35
HTR1A P08908 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
EHMT2 Q96KQ7 1/20 0.34
TNF P01375 1/20 0.34
LITAF Q99732 1/20 0.34
PDCD1LG2 Q9BQ51 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774216 0.80 SLC2A1 (0.49) KCNH2HTR1AADRA1DADRA1AADRA1B
SCHEMBL4270110 0.77 KCNH2 (0.49) KCNH2MC4RTACR1
SCHEMBL5772116 0.70 SLC2A1 (0.48) KCNH2ADORA2AKDM4EALDH1A1HTR1A
SCHEMBL4721450 0.67 CCR8 (0.53) KCNH2ADORA2AHTR1AADRA1DADRA1A
SCHEMBL5773885 0.67 KCNH2 (0.68) KCNH2
SCHEMBL3686475 0.65 KCNH2 (0.40) KCNH2KDM4EALDH1A1TACR1HTR1A
SCHEMBL13857010 0.63 FAAH (0.41) KDM4EALDH1A1
SCHEMBL3689424 0.63 HTR1A (0.44) KCNH2KDM4EALDH1A1TACR1HTR1A
SCHEMBL4718696 0.63 CCR8 (0.53) KCNH2HTR1AADRA1DADRA1AADRA1B
SCHEMBL23360169 0.62 HTR1A (0.49) ALDH1A1HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305308-B1 AMINOPIPERIDINE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2006-12-20 EP claimed