SCHEMBL3687774

SCHEMBL3687774

COc1ccc(Cl)cc1C(=O)NCCc1ccc(OC(C)(C)C(=O)O)cc1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DNMT3A Q9Y6K1 1/20 0.69
ALDH1A1 P00352 2/20 0.68
FABP2 P12104 1/20 0.68
PPARG P37231 1/20 0.68
PPARD Q03181 1/20 0.68
PPARA Q07869 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
HDAC1 Q13547 2/20 0.64
HDAC6 Q9UBN7 2/20 0.64
NLRP3 Q96P20 3/20 0.63
KDM4E B2RXH2 1/20 0.63
PKM P14618 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1154123 0.97 DNMT3A (0.66) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL1153879 0.92 ALDH1A1 (0.58) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL1153988 0.91 DNMT3A (0.60) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL1154718 0.90 DNMT3A (0.59) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL1154562 0.90 ALDH1A1 (0.56) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL5323204 0.89 PPARA (0.58) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL1154442 0.89 DNMT3A (0.58) DNMT3AALDH1A1FABP2PPARGPPARD
SCHEMBL11711852 0.89 DNMT3A (0.66) DNMT3AALDH1A1HDAC1HDAC6NLRP3
SCHEMBL1154171 0.89 DNMT3A (0.66) DNMT3AALDH1A1HDAC1HDAC6NLRP3
SCHEMBL1154002 0.89 DNMT3A (0.60) DNMT3AALDH1A1FABP2PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7795310-B2 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2010-09-14 US claimed
US-7795310-B2 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2010-09-14 US disclosed
EP-1781303-A4 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX INC (US) 2008-07-02 EP disclosed
EP-1781303-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS CombinatoRx, Incorporated (US) 2007-05-09 EP disclosed
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2006-03-30 US disclosed
WO-2006004803-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX, INCORPORATED (US) 2006-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders LIPC, PNLIP, GOT2 DNMT3A 615/4885ALDH1A1 626/4885FABP2 160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.