SCHEMBL3689633

SCHEMBL3689633

O=C(O)c1cc(-c2ccc(Cl)cc2)ccc1O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 7/20 0.72
MCL1 Q07820 6/20 0.72
HNF4A P41235 2/20 0.72
DHFR P00374 1/20 0.72
CA1 P00915 2/20 0.71
CA2 P00918 2/20 0.71
LCK P06239 2/20 0.62
ALOX5 P09917 2/20 0.59
MEN1 O00255 1/20 0.56
APP P05067 1/20 0.56
THRB P10828 1/20 0.56
RECQL P46063 1/20 0.56
BLM P54132 1/20 0.56
KMT2A Q03164 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CA12 O43570 1/20 0.53
PTGS2 P35354 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA14 Q9ULX7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29374831 0.90 ACMSD (0.88) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL18224311 0.90 ACMSD (0.88) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL29904854 0.88 ACMSD (0.83) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL2771723 0.88 ACMSD (0.83) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL22206257 0.86 ACMSD (0.80) ACMSDMCL1HNF4ADHFRCA1
Methane SCHEMBL28165586 0.86 ACMSD (0.80) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL23143193 0.84 ACMSD (1.00) ACMSDMCL1HNF4ADHFRLCK
SCHEMBL1898000 0.84 ACMSD (0.78) ACMSDMCL1HNF4ADHFRCA1
SCHEMBL9273036 0.84 ACMSD (1.00) ACMSDMCL1HNF4ADHFRLCK
SCHEMBL29759663 0.84 ACMSD (1.00) ACMSDMCL1HNF4ADHFRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7795310-B2 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2010-09-14 US disclosed
EP-1781303-A4 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX INC (US) 2008-07-02 EP disclosed
CN-101010083-A Methods and reagents for the treatment of metabolic disorders COMBINATORX INC (US) 2007-08-01 CN disclosed
EP-1781303-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS CombinatoRx, Incorporated (US) 2007-05-09 EP disclosed
CN-1867340-A Topical use of halosalicylic acid derivatives AVON PROD INC (US) 2006-11-22 CN disclosed
EP-1694337-A2 TOPICAL USE OF HALOSALICYLIC ACID DERIVATIVES AVON PRODUCTS, INC. (US) 2006-08-30 EP disclosed
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2006-03-30 US disclosed
WO-2006004803-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX, INCORPORATED (US) 2006-01-12 WO disclosed
WO-2005058230-A2 TOPICAL USE OF HALOSALICYLIC ACID DERIVATIVES AVON PRODUCTS, INC. (US) 2005-06-30 WO disclosed
US-20050136015-A1 Topical use of halosalicylic acid derivatives AVON PRODUCTS, INC. 2005-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050136015-A1 Topical use of halosalicylic acid derivatives NACA, TYR, PRKDC ACMSD 1718/4885MCL1 729/4885HNF4A 3980/4885
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders LIPC, PNLIP, GOT2 ACMSD 3350/4885MCL1 3721/4885HNF4A 116/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.