SCHEMBL3690604

SCHEMBL3690604

COc1cccc2c(C(O)CN3C4CCC3CC(NCc3cc5ccccc5o3)C4)ccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 3/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
HTR1A P08908 4/20 0.35
DRD2 P14416 3/20 0.35
HTR2B P41595 3/20 0.35
KCNH2 Q12809 4/20 0.34
CYP3A4 P08684 1/20 0.34
HTR3A P46098 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
CXCR6 O00574 1/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777778 0.88 SLC2A1 (0.47) SLC2A1HTR1ADRD2HTR2BKCNH2
SCHEMBL3698321 0.86 HCRTR1 (0.35) HCRTR1HCRTR2HTR1ADRD2HTR2B
SCHEMBL3690599 0.85 KCNH2 (0.50) SLC2A1KCNH2CYP3A4KDM4EMEN1
SCHEMBL3697149 0.78 HTR1A (0.35) HTR1AHTR2BALDH1A1ADRA1DADRA1A
SCHEMBL5778069 0.77 MEN1 (0.38) SLC2A1HTR1ADRD2HTR2BKCNH2
SCHEMBL3694555 0.76 HTR1A (0.33) HTR1AADRA1DADRA1AADRA1BSLC6A4
SCHEMBL4275508 0.72 KCNH2 (0.65) SLC2A1KCNH2
SCHEMBL3691027 0.72 CYP2D6 (0.33) HTR1AKCNH2HTR3ACYP2C19ADRA1D
SCHEMBL5652075 0.71 CCR8 (0.45) SLC2A1DRD2HTR2BKCNH2CYP3A4
SCHEMBL13145896 0.71 KCNH2 (0.48) SLC2A1DRD2HTR2BKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed