SCHEMBL3690899

SCHEMBL3690899

CCOc1ccc(C=CC(=O)O)cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.80
ALDH1A1 P00352 2/20 0.77
HPGD P15428 2/20 0.77
ALOX15 P16050 1/20 0.77
MAPK1 P28482 1/20 0.77
SMN1; SMN2 Q16637 1/20 0.77
HSD17B10 Q99714 1/20 0.77
MAPT P10636 2/20 0.74
NPC1 O15118 1/20 0.74
RAB9A P51151 1/20 0.74
KMT2A Q03164 3/20 0.73
SNCA P37840 2/20 0.73
GAA P10253 1/20 0.73
LMNA P02545 2/20 0.70
POLB P06746 1/20 0.70
ACHE P22303 3/20 0.66
FDPS P14324 3/20 0.65
CA12 O43570 1/20 0.64
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30966315 1.00 KDM4E (0.80) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL3690896 1.00 KDM4E (0.80) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL3688296 0.94 KDM4E (0.77) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL3688297 0.94 KDM4E (0.77) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL30739528 0.92 KDM4E (0.84) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL4623922 0.92 KDM4E (0.84) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL7247313 0.92 KDM4E (0.84) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL14229893 0.90 KDM4E (0.86) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL7966747 0.89 KDM4E (0.74) KDM4EALDH1A1HPGDALOX15MAPK1
SCHEMBL7966753 0.89 KDM4E (0.74) KDM4EALDH1A1HPGDALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113801022-A Ferulic acid eugenol and isoeugenol heterozygote and application thereof 贵州大学 2021-12-17 CN claimed
CN-118266572-A Application of 3-methoxyphenyl-2-acrylic compound as bitter taste inhibitor 华南理工大学 2024-07-02 CN disclosed
US-7795310-B2 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2010-09-14 US disclosed
EP-1781303-A4 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX INC (US) 2008-07-02 EP disclosed
EP-1781303-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS CombinatoRx, Incorporated (US) 2007-05-09 EP disclosed
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders COMBINATORX, INC. (US) 2006-03-30 US disclosed
WO-2006004803-A1 METHODS AND REAGENTS FOR THE TREATMENT OF METABOLIC DISORDERS COMBINATORX, INCORPORATED (US) 2006-01-12 WO disclosed
US-5559109-A Method of treating a PAF-mediated pathology or for treating or preventing psoriasis, nephritis, asthma or shock by administering a PAF antagonist SANKKO COMPANY, LIMITED (JP) 1996-09-24 US disclosed
US-5556852-A PLATELET ACTIVATING FACTOR ANTAGONISTS SANKYO COMPANY, LIMITED (JP) 1996-09-17 US disclosed
EP-0395446-B1 N-acryloylpiperazine derivatives, their preparation and their use as paf antagonists SANKYO CO (JP) 1995-03-01 EP disclosed
US-5369106-A N-acryloylpiperazine derivatives, their preparation and their use of PAF antagonists SANKYO COMPANY, LIMITED (JP) 1994-11-29 US disclosed
US-5192766-A Platelet activating factor antagonist SANKYO COMPANY, LIMITED (JP) 1993-03-09 US disclosed
EP-0395446-A2 N-acryloylpiperazine derivatives, their preparation and their use as paf antagonists Sankyo Company Limited (JP) 1990-10-31 EP disclosed
US-4337270-A ANTIALLERGENS; ANTIANAPHYLACTIC AGENTS HISAMITSU PHARMACEUTICAL CO., INC. (JP) 1982-06-29 US disclosed
US-4247597-A Electroscopic carrier particles having a carboxylic acid surface treatment PITNEY BOWES, INC. (US) 1981-01-27 US disclosed
US-4026896-A ANTIALLERGENS KISSEI YAKUHIN KOGYO KABUSHIKI KAISHA (KISSEI PHARMACEUTICAL CO. LTD.) (JA) 1977-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060069161-A1 Methods and reagents for the treatment of metabolic disorders LIPC, PNLIP, GOT2 KDM4E 3045/4885ALDH1A1 626/4885HPGD 1593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.