SCHEMBL3705293

SCHEMBL3705293

CN(Cc1cc(S(=O)(=O)c2cccnc2)n(-c2cc(F)ccc2Cl)n1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.39
SLC6A4 P31645 8/20 0.39
HTR2A P28223 1/20 0.39
NAMPT P43490 4/20 0.34
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
RORC P51449 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
FPR1 P21462 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.31
PTGER2 P43116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700851 0.92 HTR2C (0.39) HTR2CSLC6A4HTR2ARORC
SCHEMBL3693157 0.92 HTR2C (0.43) HTR2CSLC6A4HTR2ANAMPTABCC9
SCHEMBL3697102 0.89 HTR2C (0.41) HTR2CSLC6A4HTR2ANAMPT
SCHEMBL4566347 0.89 HTR2C (0.39) HTR2CSLC6A4HTR2AABCC9ABCC8
SCHEMBL4131429 0.88 KEAP1 (0.36) NAMPTALDH1A1KEAP1NFE2L2LMNA
SCHEMBL3808572 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2ANAMPTABCC9
SCHEMBL3699812 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2AABCC9ABCC8
SCHEMBL3695801 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2ANAMPTABCC9
SCHEMBL3701316 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2ANAMPTABCC9
SCHEMBL3705296 0.83 NAMPT (0.34) NAMPTABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed