SCHEMBL3699787

SCHEMBL3699787

O=C(NNOC(=O)c1nc2c(C(F)(F)F)cc(-c3ccco3)cn2c1Cl)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CFTR P13569 2/20 0.38
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
POLB P06746 3/20 0.37
ADORA3 P0DMS8 1/20 0.36
KAT6A Q92794 4/20 0.35
SCD5 Q86SK9 2/20 0.35
HDAC2 Q92769 1/20 0.35
RAB9A P51151 2/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
CYP2C8 P10632 2/20 0.34
CYP2B6 P20813 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSD17B10 Q99714 2/20 0.34
ESR1 P03372 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1583743 0.85 CFTR (0.53) PKMRXFP1CFTRALDH1A1KDM4E
SCHEMBL1583694 0.82 KDM4E (0.41) PKMRXFP1CFTRALDH1A1KDM4E
SCHEMBL3699785 0.82 ADORA3 (0.39) PKMRXFP1CFTRALDH1A1KDM4E
SCHEMBL3690164 0.81 ALDH1A1 (0.47) PKMCFTRALDH1A1KDM4EPOLB
SCHEMBL3696233 0.80 PKM (0.49) PKMRXFP1ALDH1A1KDM4EPOLB
SCHEMBL3684339 0.79 ALDH1A1 (0.48) PKMRXFP1ALDH1A1KDM4EPOLB
SCHEMBL3703771 0.78 SCD5 (0.47) PKMRXFP1ADORA3SCD5CYP2C8
SCHEMBL7490436 0.77 ALDH1A1 (0.48) PKMRXFP1ALDH1A1KDM4EPOLB
SCHEMBL3702560 0.77 ADORA2A (0.46) PKMRXFP1ALDH1A1ADORA3RAB9A
SCHEMBL7495802 0.77 CACNA1B (0.48) PKMRXFP1ALDH1A1KDM4ESCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections OAT, HAVCR2, CPS1 PKM 2286/4885RXFP1 4676/4885CFTR 2042/4885
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections OAT, HAVCR2, CPS1 PKM 2286/4885RXFP1 4676/4885CFTR 2042/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.