SCHEMBL3700701

SCHEMBL3700701

Cc1ccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2cccc(F)c2C)cn1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
SCN9A Q15858 3/20 0.32
SCN5A Q14524 1/20 0.32
PTGS2 P35354 2/20 0.31
NAMPT P43490 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703103 0.95 NAMPT (0.33) NAMPT
SCHEMBL3700610 0.94 SLC16A3 (0.33) PTGS2NAMPTHTR2AHTR2CKCNH2
SCHEMBL3697675 0.92 ALDH1A1 (0.35) RXRAGRIN1GRIN2BSCN9ASCN5A
SCHEMBL3699813 0.90 ABCC9 (0.34) NAMPT
SCHEMBL3688572 0.90 RIPK1 (0.34) RXRAGRIN1GRIN2B
SCHEMBL3698342 0.88 NAMPT (0.31) PTGS2NAMPT
SCHEMBL3696613 0.87 SLC16A3 (0.37)
SCHEMBL4125819 0.87 PTGS2 (0.33) RXRAGRIN1GRIN2BSCN9ASCN5A
SCHEMBL4200027 0.87 MEN1 (0.32)
Fumaric Acid SCHEMBL3695034 0.86 NAMPT (0.30) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed