SCHEMBL3700610

SCHEMBL3700610

Cc1ccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2ccccc2F)cn1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 6/20 0.33
SLC16A1 P53985 6/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
KCNH2 Q12809 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
ESR1 P03372 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NTRK1 P04629 1/20 0.31
NAMPT P43490 2/20 0.31
PTGS2 P35354 2/20 0.31
CTSA P10619 2/20 0.31
CYP3A4 P08684 1/20 0.31
SPR P35270 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700701 0.94 RXRA (0.32) HTR2AHTR2CKCNH2NAMPTPTGS2
Fumaric Acid SCHEMBL3695034 0.91 NAMPT (0.30) NAMPT
SCHEMBL3698589 0.91 ALDH1A1 (0.38) SLC16A3SLC16A1HTR2AHTR2CKCNH2
SCHEMBL3698342 0.91 NAMPT (0.31) NAMPTPTGS2
SCHEMBL3805211 0.90 TAS2R14 (0.38) SLC16A3SLC16A1HTR2AHTR2CKCNH2
SCHEMBL3696613 0.90 SLC16A3 (0.37) SLC16A3SLC16A1ALDH1A1
SCHEMBL3703103 0.90 NAMPT (0.33) ABCC9ABCC8KCNJ11KCNJ8NAMPT
SCHEMBL3808574 0.89 ABCC9 (0.35) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL3688572 0.89 RIPK1 (0.34) SLC16A3SLC16A1
SCHEMBL4130428 0.87 SLC16A3 (0.34) SLC16A3SLC16A1HTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed