SCHEMBL3702497

SCHEMBL3702497

CC(C)(C)C(Cc1cccc(NC(=O)C(c2ccc(Cn3nc(-c4ccccc4)oc3=O)cc2)C2CCCC2)c1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGES O14684 5/20 0.44
HTR1E P28566 3/20 0.40
S1PR3 Q99500 3/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.39
ACKR3 P25106 3/20 0.38
PTGS2 P35354 5/20 0.36
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
NPY1R P25929 1/20 0.35
CCR3 P51677 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3702669 0.86 PTGES (0.60) PTGESHTR1ES1PR3MEN1LMNA
SCHEMBL1083357 0.86 PTGS2 (0.49) PTGESPTGS2
SCHEMBL1177701 0.85 PTGES (0.49) PTGESHTR1ES1PR3MEN1LMNA
SCHEMBL7601841 0.85 PTGES (0.52) PTGESHTR1ES1PR3MEN1LMNA
SCHEMBL3701755 0.81 LMNA (0.42) PTGESHTR1ES1PR3MEN1LMNA
SCHEMBL3692778 0.80 PTGES (0.44) PTGESHTR1ES1PR3MEN1LMNA
SCHEMBL12871550 0.79 GRIN1 (0.47) FAAHMGLL
SCHEMBL1178321 0.79 PTGES (0.46) PTGESHTR1ES1PR3MEN1LMNA
Bicarbonate SCHEMBL3693730 0.78 BDKRB2 (0.44) HTR1ES1PR3MEN1LMNAKMT2A
SCHEMBL1177898 0.77 CYP1A2 (0.51) PTGESHTR1ES1PR3MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed