SCHEMBL3705296

SCHEMBL3705296

CC(C)(C)CN(Cc1cc(S(=O)(=O)c2cccnc2)n(-c2cc(F)ccc2Cl)n1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.34
TP53 P04637 2/20 0.33
LMNA P02545 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
PTGER2 P43116 6/20 0.33
KEAP1 Q14145 2/20 0.32
NFE2L2 Q16236 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
MAPT P10636 3/20 0.32
ALDH1A1 P00352 2/20 0.32
FPR1 P21462 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700854 0.92 NAMPT (0.30) NAMPT
SCHEMBL3693161 0.92 NAMPT (0.36) NAMPTTP53LMNATAS2R14ABCC9
SCHEMBL3697103 0.89 PRCP (0.33) PTGDR2
SCHEMBL4566348 0.89 PTGER2 (0.33) TAS2R14ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4131429 0.88 KEAP1 (0.36) NAMPTTP53LMNATAS2R14PTGER2
SCHEMBL3808574 0.87 ABCC9 (0.35) NAMPTTP53ABCC9ABCC8KCNJ11
SCHEMBL3695804 0.85 ABCC9 (0.34) NAMPTTP53ABCC9ABCC8KCNJ11
SCHEMBL3699813 0.85 ABCC9 (0.34) NAMPTTP53ABCC9ABCC8KCNJ11
SCHEMBL3701318 0.85 NAMPT (0.36) NAMPTTP53LMNAABCC9ABCC8
Fumaric Acid SCHEMBL3702665 0.83 NAMPT (0.36) NAMPTABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed